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A-3 hydrochloride

Glpbio
Catalog No:GC60037-10mM (in 1mL DMSO) CAS No.:78957-85-4 MDLNo:C12H14Cl2N2O2S Brand:Glpbio purity: 特性: Purpose:A-3 hydrochloride 是靶向多种激酶 (kinase) 的强效、细胞渗透的、可逆的、ATP 竞争性的非选择性拮抗剂。A-3 hydrochloride 是针对 PKA (Ki=4.3 µM),酪蛋白激酶 II (Ki=5.1 µM) 和肌球蛋白轻链激酶 (MLCK) (Ki=7.4 µM) 的抑制剂。A-3 hydrochloride 还抑制 PKC 和酪蛋白激酶 I 的活性,Ki 分别为 47 µM 和 80 µM。DMSO: 125 mg/mL (389.14 mM; Need ultrasonic)
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Product Overview
Product Name A-3 hydrochloride
CAS78957-85-4
MW321.22
MDLC12H14Cl2N2O2S
Storage conditionPowder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
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